5-HT Receptor


5-HT receptors (5-hydroxytryptamine receptors,The serotonin receptors) are a group of G protein-coupled receptors (GPCRs) and ligand-gated ion channels (LGICs) found in the central and peripheral nervous systems. They mediate both excitatory and inhibitory neurotransmission. The serotonin receptors are activated by the neurotransmitter serotonin, which acts as their natural ligand.

  • EMD 386088 hydrochloride EI1076

    EMD 386088 hydrochloride是活性的 5-HT6 激动剂。

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  • EMD 281014 hydrochloride EI1075

    EMD 281014 hydrochloride是选择性 5-HT2A 拮抗剂。

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  • Eltoprazine hydrochloride EI1074

    Eltoprazine hydrochloride是5-HT1 受体激动剂/部分激动剂。

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  • DV 7028 hydrochloride EI1042

    DV 7028 hydrochloride是选择性 5-HT2A 拮抗剂,抗血栓剂。

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  • DR 4485 hydrochloride EI1038

    DR 4485 hydrochloride是高亲和性选择性 5-HT7 拮抗剂, 口服有效。

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  • EMD 386088 hydrochloride EI1076

    EMD 386088 hydrochloride是活性的 5-HT6 激动剂。

    More
  • EMD 281014 hydrochloride EI1075

    EMD 281014 hydrochloride是选择性 5-HT2A 拮抗剂。

    More
  • Eltoprazine hydrochloride EI1074

    Eltoprazine hydrochloride是5-HT1 受体激动剂/部分激动剂。

    More
  • DV 7028 hydrochloride EI1042

    DV 7028 hydrochloride是选择性 5-HT2A 拮抗剂,抗血栓剂。

    More
  • DR 4485 hydrochloride EI1038

    DR 4485 hydrochloride是高亲和性选择性 5-HT7 拮抗剂, 口服有效。

    More
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